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1-Azakenpaullone (9-Bromo-7,12-dihydropyridoazepinoindol-6(5H)-one)

1-Azakenpaullone (9-Bromo-7,12-dihydropyridoazepinoindol-6(5H)-one)

Cat no: 044431

Supplier: United States Biological
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Potent and ATP-competitive GSK-3beta (glycogen synthase kinase-3beta) inhibitor (IC50 = 18 nM). Storage and Stability: Short-term Storage: +4 degrees C Long-term Storage: -20 degrees C Stable for at least 2 years after receipt when stored at -20 degrees C.
Catalogue number: 044431
Size: 1mg
Purity: >98% (NMR)
Alternative names: 9-Bromo-7,12-dihydropyridoazepinoindol-6(5H)-one
References: Product Reference: ?1-Azakenpaullone is a selective inhibitor of glycogen synthase kinase-3 beta: C. Kunick, et al.; Bioorg. Med. Chem. Lett.14, 413 (2004) ?Studying the mechanism that enables paullones to selectively inhibit glycogen synthase kinase 3 rather than cyclin-dependent kinase 5 by molecular dynamics simulations and free-energy calculations: Q. Chen, et al.; J. Mol. Model. Epub ahead of print (2010) ?

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