DPCPX is a potent and very selective A1-adenosine receptor antagonist, with a Ki of 0.46 nM for A1 receptors in rat whole-brain membranes. Its 740-fold A1-selectivity is the highest reported for an adenosine antagonist.
Melting Point: 191-194 degrees C
Solubility: DMSO (3.6 mg/ml), Ethanol (4 mg/ml), 0.1N Sodium Hydroxide (2 mg/ml)
Storage and Stability:
May be stored at RT for short-term only. Long-term storage is recommended at -20 degrees C. For maximum recovery of product, centrifuge the original vial prior to removing the cap.