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IC87114, PI3K Inhibitor (2-[6-Amino-9H-purin-9-yl)methyl]-5-methyl-3-(2-methylphenyl)-4(3H)-quinazolinone)

IC87114, PI3K Inhibitor (2-[6-Amino-9H-purin-9-yl)methyl]-5-methyl-3-(2-methylphenyl)-4(3H)-quinazolinone)

Cat no: I0504

Supplier: United States Biological
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Cell-permeable. A potent, ATP-competitive and selective inhibitor of PI 3-K isoform p110e (IC?? =60nM). Inhibits p110a and p110b only at higher concentrations (>1uM). IC87114 does not inhibit other PIK-related kinases such as ATM, ATR, DNA-PK, and mTOR even at concentrations up to 100uM. Solubility: DMSO Molecular Weight: ~397.43 Storage and Stability: Lyophilized powder may be stored at -20 degrees C. Stable for 12 months at -20 degrees C. Reconstitute with DMSO. Aliquot to avoid repeated freezing and thawing. Store at -20 degrees C. For maximum recovery of product, centrifuge the original vial after thawing and prior to removing the cap. Further dilutions can be made in assay buffer.
Catalogue number: I0504
Size: 1mg
Form: Supplied as a white to off-white solid.
Purity: ~95% (HPLC)
References: 1. Chaussade, C., et al. (2007). Biochem. J. 404, 449.

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