A selective inhibitor of protein kinase C or cyclic-nucleotide-dependent protein kinases. Form: Light Yellow Powder
A selective inhibitor of dopamine uptake. An antidepressant of the aminoketone class; aid in smoking cessation. Form: White Solid Melting Point: 153-157...
A selective inhibitor of dopamine uptake. An antidepressant of the aminoketone class; aid in smoking cessation. Form: White Solid Melting Point: 153-155...
A selective inhibitor of BCL-2, in small cell lung cancer. ABT-737 induced dramatic regressions in tumors derived from some SCLC cell lines. Form: Yellow...
A selective inhibitor of BCL-2, in small cell lung cancer. ABT-737 induced dramatic regressions in tumors derived from some SCLC cell lines. Form: Yellow...
A selective inhibitor of ALK5 kinase.
A selective estrogen receptor modulator. Form: Off-White Solid Melting Point: 135-144 degrees C Solubility: Acetone, Dichloromethane, Methanol
A selective E-prostanoid receptor subtype 1 (EP1) receptor antagonist which shows antihypertensive effects. Form: Off-White Solid Melting Point: 112-114...
A selective EP1 prostanoid receptor antagonist that attenuates prostaglandin E2-induced neuronal cell death in vitro and slows tumor growth in vivo. Its...
A selective dopamine D2-receptor antagonist with dopamine autoreceptor agonist activity. Antipsychotic. Form: Off-White Solid Melting Point: 138-140 degrees...
A selective D4 dopamine antagonist that exhibits low affinity at other monoamine receptors (Ki > 2000 nM). Induces c-fos gene expression in medial prefrontal...
A selective cyclooxygenase-2 (COX-2) inhibitor. Anti-inflammatory. Used in treatment of familial adenomatous polyposis. Form: White to Pale Yellow Solid...
A selective class II (IIa) histone deacetylase (HDAC II) inhibitor. It exhibits tissue-selective inhibition between members of class II acetylases in vivo,...
A selective cAMP phosphodiesterase (PDE-3) inhibitor with positive inotropic and vasodilatory activity. Cardiotonic. Form: Brown Solid Melting Point: >240...
A selective and potent non-peptide angiotensin II type 2 (AT2) receptor antagonist. Potential treatment of cardiac hypertrophy as blockage of AT2 receptor...
A selective acetylcholinesterase inhibitor. Form: Off-White Solid Melting Point: 183-185 degrees C Solubility: Chloroform, Dichloromethane
A selective A2A receptor agonist. Form: White to Off-White Solid Melting Point: 204-206 degrees C Solubility: DMSO, Methanol
A selective A2A receptor agonist. Form: Off-White Solid Melting Point: 167-174 degrees C Solubility: Water
A selective A2A adenosine receptor agonist in myocardial imaging. Form: Pale Beige Solid Melting Point: 200-205 degrees C (dec.) Solubility: DMSO, Methanol
A selective 5-HT4 receptor agonist. Gastroprokinetic. Form: White Solid Melting Point: 112-114 degrees C Solubility: DMSO, Methanol