A selective, non-peptide antagonist of corticotropin releasing factor receptors (CRF1). It blocks CRF-induced adenylate cyclase activation and attenuates...
A selective, competitive HMG-CoA reductase inhibitor. The only drug in its class specfically indicated for lowering both elevated LDL-cholesterol and...
A selective d6 desaturase inhibitor (IC50 = 0.2uM in vitro). Displays selectivity over d5 and d9 desaturases (IC50 values are >200 microM in vitro). It...
A selective tyrosine kinase inhibitor. Form: Light Yellow Solid Solubility: Chloroform, Dichloromethane, Ethyl Acetate
A selective serotonin reuptake inhibitor (SSRI). Used as an antidepressant. Form: White Solid Melting Point: 126-129 degrees C Solubility: Chloroform
A selective serotonin reuptake inhibitor (SSRI) used as an anti-depressant. Form: Colourless Oil Solubility: Chloroform, Dichloromethane, Petroleum Ether
A selective pre-emergence herbicide. Form: Pale Yellow Oil Solubility: Chloroform, Methanol
A selective NaV1.8 sodium channel blocker, reduces behavioral measures of chronic pain. Form: White Solid Melting Point: 128-130 degrees C Solubility: DMSO,...
A selective muscarinic receptor stimulant, used to treat cerebral palsy. Form: White Solid Melting Point: 187-190 degrees C Solubility: Methanol
A selective leukotriene D4-receptor antagonist. Used as an antiasthmatic. Form: Pale Beige Solid Melting Point: 65-67 degrees C Solubility: Chloroform, Methanol
A selective labeled cyclooxygenase-2 (COX-2) inhibitor. Use as an anti-inflammatory, analgesic. Form: White Solid Melting Point: 208-210 degrees C...
A selective inhibitor of protein kinase C or cyclic-nucleotide-dependent protein kinases. Form: Light Yellow Powder
A selective inhibitor of dopamine uptake. An antidepressant of the aminoketone class; aid in smoking cessation. Form: White Solid Melting Point: 153-157...
A selective inhibitor of dopamine uptake. An antidepressant of the aminoketone class; aid in smoking cessation. Form: White Solid Melting Point: 153-155...
A selective inhibitor of BCL-2, in small cell lung cancer. ABT-737 induced dramatic regressions in tumors derived from some SCLC cell lines. Form: Yellow...
A selective inhibitor of BCL-2, in small cell lung cancer. ABT-737 induced dramatic regressions in tumors derived from some SCLC cell lines. Form: Yellow...
A selective inhibitor of ALK5 kinase.
A selective estrogen receptor modulator. Form: Off-White Solid Melting Point: 135-144 degrees C Solubility: Acetone, Dichloromethane, Methanol
A selective E-prostanoid receptor subtype 1 (EP1) receptor antagonist which shows antihypertensive effects. Form: Off-White Solid Melting Point: 112-114...
A selective EP1 prostanoid receptor antagonist that attenuates prostaglandin E2-induced neuronal cell death in vitro and slows tumor growth in vivo. Its...