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Centrally acting a-adrenoceptor agonist. Antihypertensive. Form: White Solid Melting Point: 208-211 degrees C Solubility: Unstable in methanol solution
Centrally acting myorelaxant; formerly used as an antispasmodic and uricosuric. Used as a tool for assessing hepatic cytochrome P-450 activity in rodents....
Centrally acting muscle relaxant with expectorant properties. Form: White Solid Melting Point: 79-81 degrees C Solubility: Dichloromethane, Ethyl Acetate,...
CENPH, belongs to the centromere protein H family. This protein is component of the CENPA-NAC (nucleosome-associated) complex that plays a central role in...
Cell-permeable. YM-201636 is a selective inhibitor of phosphoinositide kinase (PIK) PIKfyve (IC503nM). It inhibits p110a at higher concentration (IC50=3uM)....
Cell-permeable. Salermide is an inhibitor of SIRT1 and SIRT2. In vitro, Salermide has a stronger inhibitory effect on SIRT2 than on SIRT1. It induces massive...
Cell-permeable. LDN-57444 is a potent, reversible, competitive and active site-directed inhibitor of UCHL1 (Ki = 0.4uM). Decreases proteasome activity and...
Cell-permeable. An anti-diabetic agent. ATP-sensitive potassium channel (KATP) blocker. Inhibits KATP currents in the pancreatic beta cells causing an...
Cell-permeable. A thiazolidinedione (TZD) derivative that acts as a selective peroxisome proliferator-activated receptor gamma (PPARg) agonist (EC50 =...
Cell-permeable. A potent protein kinase C (PKC) inhibitor (IC50 = 7.9nM). In vitro, discriminates between Ca2+- dependent and -independent isoforms of PKC;...
Cell-permeable, non-selective broad-spectrum caspase inhibitor. Binds irreversibly to the catalytic site of caspase proteases. The peptide is O-methylated in...
Cellobionic acid is produced by ozonization of Cellobiose. Cellobionic acid was not a good substrate for b-Glucosidase. The lactonized carboxyl group...
Cell permeable, specific p38 MAP kinase inhibitor. Binds to the ATP binding site of p38 MAP kinase. T cell proliferation inhibitor. IL-2 production...
Cell permeable, potent, selective, non-transition state and non-competitive gamma-secretase inhibitor. Notch processing inhibitor. Only weakly affects...
Cell permeable, non-fluorescent F-actin probe. Potent inducer of actin polymerization and stabilization. Competes with phallotoxins for actin binding....
Cell permeable, highly potent inhibitor of gamma-secretase (IC50 = 0.06nM). Storage and Stability: Short-term Storage: +4 degrees C Long-term Storage: -20...
Cell permeable, competitive, non-specific cAMP and cGMP phosphodiesterase inhibitor. Increases cAMP levels that activate PKA, leading to decreased...
Cell permeable superoxide dismutase (SOD) mimetic. Potent inhibitor of peroxynitrite-induced oxidative reactions (peroxynitrite scavenger), but not a...
Cell permeable superoxide dismutase (SOD) mimetic. Peroxynitrite scavenger. Displays a protective effect against H2O2 mediated injury. Neuroprotective....
Cell permeable steroidal alkaloid. Specific sonic hedgehog signaling (Shh) pathway inhibitor. Directly interacts/inhibits Smo (smoothened). Teratogenic and...
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